Molecule Details
| General Information of the Molecule | ||||
|---|---|---|---|---|
| Name |
Norepinephrine transporter (NET)
|
|||
| Synonyms |
Solute carrier family 6 member 2; Sodium-dependent noradrenaline transporter; SLC6A2; NET1; NET; NAT1
|
|||
| Gene Name |
SLC6A2
|
|||
| Gene ID | ||||
| Sequence |
MLLARMNPQVQPENNGADTGPEQPLRARKTAELLVVKERNGVQCLLAPRDGDAQPRETWG
KKIDFLLSVVGFAVDLANVWRFPYLCYKNGGGAFLIPYTLFLIIAGMPLFYMELALGQYN REGAATVWKICPFFKGVGYAVILIALYVGFYYNVIIAWSLYYLFSSFTLNLPWTDCGHTW NSPNCTDPKLLNGSVLGNHTKYSKYKFTPAAEFYERGVLHLHESSGIHDIGLPQWQLLLC LMVVVIVLYFSLWKGVKTSGKVVWITATLPYFVLFVLLVHGVTLPGASNGINAYLHIDFY RLKEATVWIDAATQIFFSLGAGFGVLIAFASYNKFDNNCYRDALLTSSINCITSFVSGFA IFSILGYMAHEHKVNIEDVATEGAGLVFILYPEAISTLSGSTFWAVVFFVMLLALGLDSS MGGMEAVITGLADDFQVLKRHRKLFTFGVTFSTFLLALFCITKGGIYVLTLLDTFAAGTS ILFAVLMEAIGVSWFYGVDRFSNDIQQMMGFRPGLYWRLCWKFVSPAFLLFVVVVSIINF KPLTYDDYIFPPWANWVGWGIALSSMVLVPIYVIYKFLSTQGSLWERLAYGITPENEHHL VAQRDIRQFQLQHWLAI Click to Show/Hide
|
|||
| Function |
Amine transporter. Terminates the action of noradrenaline by its high affinity sodium-dependent reuptake into presynaptic terminals.
Click to Show/Hide
|
|||
| Uniprot ID | ||||
| Pfam | ||||
| TTD ID | ||||
| VARIDT ID | ||||
| Drug(s) of This Target | ||||
|---|---|---|---|---|
| 1 | Bupropion | Drug Info | Approved | Nicotine use disorder |
| 2 | Diethylpropion | Drug Info | Approved | Obesity |
| 3 | Duloxetine | Drug Info | Approved | Depression |
| 4 | Imipramine | Drug Info | Approved | Depression |
| 5 | Paracetamol | Drug Info | Approved | Pain |
| 6 | Tapentadol | Drug Info | Approved | Acute pain |
| 7 | Venlafaxine | Drug Info | Approved | Depression |